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CCZ01048

Product Specifications

Target

Melanocortin Receptor

Related Pathways

Neuroscience|||GPCR/G Protein

Bioactivity

CCZ01048, an analogue of ?-melanocyte-stimulating hormone (?-MSH), demonstrates a high binding affinity for the melanocortin 1 receptor (MC1R), with a Ki of 0.31 nM. It rapidly internalizes into B16F10 melanoma cells and exhibits notable in vivo stability, making it a promising candidate for PET imaging of malignant melanoma [1].

Molecular Formula

C71H105N21O16

Molecular Weight

1508.72

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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