TAT-cyclo-CLLFVY TFA
Product Specifications
Target
HIF/HIF Prolyl-Hydroxylase
Related Pathways
Metabolism|||Chromatin/Epigenetic
Bioactivity
TAT-cyclo-CLLFVY TFA is a cyclic peptide inhibitor targeting HIF-1 heterodimerization to mitigate hypoxia signaling within cancer cells. It effectively disrupts the protein-protein interaction between HIF-1? and HIF-1?, with an inhibitory concentration (IC 50) of 1.3 ?M [1].
Molecular Formula
C113H189F3N42O26S2
Molecular Weight
2673.1
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Product Datasheet
https://www.targetmol.com/attachment/DataSheet/64416151915987135/T75943
Available Sizes
Curated Selection
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