PL-017 TFA
Product Specifications
Target
Opioid Receptor
Related Pathways
Neuroscience, GPCR/G Protein, Endocrinology/Hormones
Bioactivity
PL-017 TFA, a potent and selective μ-opioid receptor agonist, displays significant affinity with an IC50 of 5.5 nM for 125I-FK 33,824 binding to the μ-site. This compound is effective in producing long-lasting, reversible analgesia in rats [1].
Molecular Formula
C31H38F3N5O7
Molecular Weight
649.66
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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