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PL-017 TFA

Product Specifications

Target

Opioid Receptor

Related Pathways

Neuroscience, GPCR/G Protein, Endocrinology/Hormones

Bioactivity

PL-017 TFA, a potent and selective μ-opioid receptor agonist, displays significant affinity with an IC50 of 5.5 nM for 125I-FK 33,824 binding to the μ-site. This compound is effective in producing long-lasting, reversible analgesia in rats [1].

Molecular Formula

C31H38F3N5O7

Molecular Weight

649.66

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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