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UFP-101 TFA

Product Specifications

Target

Opioid Receptor

Related Pathways

GPCR/G Protein, Endocrinology/Hormones, Neuroscience

Bioactivity

UFP-101 TFA is a potent, selective, and competitive N/OFQ peptide (NOP) receptor antagonist with a pKi value of 10.24, showing over 3000-fold selectivity against δ, μ, and κ opioid receptors, and exhibits antidepressant-like effects [1] [2].

Molecular Formula

C84H139F3N32O23

Molecular Weight

2022.19

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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