UFP-101 TFA
Product Specifications
Target
Opioid Receptor
Related Pathways
GPCR/G Protein, Endocrinology/Hormones, Neuroscience
Bioactivity
UFP-101 TFA is a potent, selective, and competitive N/OFQ peptide (NOP) receptor antagonist with a pKi value of 10.24, showing over 3000-fold selectivity against δ, μ, and κ opioid receptors, and exhibits antidepressant-like effects [1] [2].
Molecular Formula
C84H139F3N32O23
Molecular Weight
2022.19
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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