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ANQ-11125 TFA

Product Specifications

Target

Motilin Receptor

Related Pathways

GPCR/G Protein

Bioactivity

ANQ-11125 TFA is a potent, selective motilin antagonist, exhibiting a pKd of 8.24. It effectively inhibits motilide-induced contractions in rabbit models, as demonstrated in vitro [1] [2].

Molecular Formula

C88H126F3N19O23

Molecular Weight

1875.05

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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