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HS014 TFA

Product Specifications

Target

Melanocortin Receptor

Related Pathways

GPCR/G Protein|||Neuroscience

Bioactivity

HS014 TFA, a potent and selective antagonist of the melanocortin-4 (MC4) receptor, exhibits K i values of 3.16, 108, 54.4, and 694 nM for the human MC4, MC1, MC3, and MC5 receptors, respectively. It effectively increases food intake in free-feeding rats [1] [2].

Molecular Formula

C73H95F3N20O19S2

Molecular Weight

1677.78

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/64416151915987045/T75853

Available Sizes

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