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Cyclosomatostatin TFA

Product Specifications

Target

Somatostatin

Related Pathways

GPCR/G Protein

Bioactivity

Cyclosomatostatin TFA, a potent somatostatin (SST) receptor antagonist, inhibits type 1 somatostatin receptor (SSTR1) signaling, reducing cell proliferation, the size of the ALDH+ cell population, and sphere-formation in colorectal cancer (CRC) cells [1].

Molecular Formula

C46H58F3N7O8

Molecular Weight

893.99

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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