Antagonist G TFA
Product Specifications
Target
Apoptosis, Vasopressin Receptor
Related Pathways
GPCR/G Protein, Apoptosis
Bioactivity
Antagonist G TFA is a potent antagonist of vasopressin and exhibits weaker antagonistic effects on GRP and Bradykinin. Additionally, this compound promotes AP-1 transcription and enhances cellular sensitivity to chemotherapy [1] [2].
Molecular Formula
C51H67F3N12O8S
Molecular Weight
1065.21
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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