[Orn5]-URP TFA
Product Specifications
Target
GPCR
Related Pathways
Endocrinology/Hormones, GPCR/G Protein
Bioactivity
[Orn5]-URP TFA acts as a potent and selective antagonist exclusively targeting the Urotensin-II receptor (UT), devoid of any agonist activity, and demonstrates a significant inhibitory efficiency with a pEC50 value of 7.24 [1] [2].
Molecular Formula
C50H63F3N10O12S2
Molecular Weight
1117.22
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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