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[Orn5]-URP TFA

Product Specifications

Target

GPCR

Related Pathways

Endocrinology/Hormones, GPCR/G Protein

Bioactivity

[Orn5]-URP TFA acts as a potent and selective antagonist exclusively targeting the Urotensin-II receptor (UT), devoid of any agonist activity, and demonstrates a significant inhibitory efficiency with a pEC50 value of 7.24 [1] [2].

Molecular Formula

C50H63F3N10O12S2

Molecular Weight

1117.22

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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