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AKTide-2T TFA

Product Specifications

Target

Akt

Related Pathways

PI3K/Akt/mTOR signaling, Cytoskeletal Signaling

Bioactivity

AKTide-2T TFA, serving as an optimal in vitro substrate for AKT, demonstrates competitive inhibition of histone H2B phosphorylation with a Ki value of 12 nM. It effectively mimics the optimal phosphorylation sequence of Akt and acts as an inhibitory peptide, distinct from the wildtype AKTide due to the absence of Thr at the S22 position [1].

Molecular Formula

C76H115F3N28O22

Molecular Weight

1829.89

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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