What is the catalog number for CALP1 TFA?

The catalog number for CALP1 TFA is T75791.

What sizes are available for CALP1 TFA?

CALP1 TFA is available in the following size(s): 5 mg, 50 mg.

How many pack sizes does CALP1 TFA come in?

CALP1 TFA is available in 2 different pack sizes.

Is CALP1 TFA in stock?

CALP1 TFA is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures CALP1 TFA?

CALP1 TFA is manufactured by Molfinity.

What is the estimated delivery time for CALP1 TFA?

Estimated delivery time for CALP1 TFA is approximately 10 business day(s), depending on your location.

CALP1 TFA

Product Specifications

Target

CaMK, Apoptosis, PDE, GluR

Related Pathways

Apoptosis, Metabolism, Neuroscience

Bioactivity

CALP1 TFA, a calmodulin (CaM) agonist with a dissociation constant (Kd) of 88 μM, selectively binds to the CaM EF-hand/Ca2+-binding site, inhibiting calcium channel opening. This action blocks calcium influx and apoptosis with an IC50 of 44.78 μM, modulates glutamate receptor channel activity, and impedes a store-operated nonselective cation channel. Additionally, CALP1 TFA enhances CaM-dependent phosphodiesterase activity, denoting its multifaceted role in modulating cellular calcium dynamics [1] [2] [3] [4].