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Apelin-17 (human, bovine) TFA

Product Specifications

Target

Apelin receptor|||HIV Protease

Related Pathways

Proteases/Proteasome|||Microbiology/Virology|||GPCR/G Protein

Bioactivity

Apelin-17 (human, bovine) TFA is an endogenous agonist of the orphan G protein-coupled receptor APJ, demonstrating affinity for human APJ receptors on HEK 293 cells with a pIC50 value of 9.02. It also blocks the entry of certain HIV-1 and HIV-2 strains into NP2/CD4 cells that express the APJ receptor [1] [2] [3].

Molecular Formula

C98H157F3N34O22S

Molecular Weight

2252.57

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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