Apelin-36 (human) TFA
Product Specifications
Target
HIV Protease, Apelin receptor
Related Pathways
Microbiology/Virology, GPCR/G Protein, Proteases/Proteasome
Bioactivity
Apelin-36 (human) TFA, an endogenous agonist of the orphan G protein-coupled receptor APJ, exhibits a potent EC50 of 20 nM and high affinity (pIC5 50 = 8.61) for human APJ receptors in HEK 293 cells. It is involved in significant cardiovascular and metabolic activities. Furthermore, Apelin-36 (human) TFA can inhibit the entry of certain HIV-1 and HIV-2 strains into NP2/CD4 cells expressing the APJ receptor. [1] [2] [3] [4]
Molecular Formula
C186H298F3N69O45S
Molecular Weight
4309.85
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog