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PKI (5-24) TFA

Product Specifications

Target

PKA

Related Pathways

Tyrosine Kinase/Adaptors

Bioactivity

PKI (5-24) TFA is a synthetic peptide inhibitor of PKA (cAMP-dependent protein kinase) with potent and competitive inhibition properties, exhibiting a K i of 2.3 nM. It corresponds to residues 5-24 of the natural heat-stable protein kinase inhibitor [1][2].

Molecular Formula

C94H148N32O31.C2HF3O2

Molecular Weight

2336.4

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/64416151911792798/T75739

Available Sizes

Curated Selection

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