BIM-26226
Product Specifications
CAS Number
136207-23-3
Target
Bombesin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
BIM-26226, a gastrin-releasing peptide, serves as a potent and selective antagonist to the bombesin receptor, effectively inhibiting BN- or GRP-stimulated amylase release with IC50 values in the nanomolar range. It is utilized in cancer research [1] [2].
Smiles
C([C@H](NC([C@@H](NC([C@@H](CC1=C(F)C(F)=C(F)C(F)=C1F)N)=O)CCC(N)=O)=O)C(N[C@H](C(N[C@H](C(N[C@@H](C(N[C@@H](CC2=CN=CN2)C(N[C@H](C(OC)=O)CC(C)C)=O)=O)C)=O)[C@H](C)C)=O)C)=O)C=3C=4C(NC3)=CC=CC4
Molecular Formula
C49H63F5N12O10
Molecular Weight
1075.09
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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