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Ubiquitination-IN-2

Product Specifications

Target

E1/E2/E3 Enzyme|||Others

Related Pathways

Others|||Ubiquitination

Bioactivity

Ubiquitination-IN-2 is a potent inhibitor of E1-E2 protein?protein interactions (PPI), exhibiting inhibitory activity with a dissociation constant (Kd) of 0.72 ?M for the ubiquitin E1 (Uba1) enzyme. By blocking the transfer of ubiquitin from E1 to E2, Ubiquitination-IN-2 serves as a valuable tool in cancer research [1].

Molecular Formula

C93H173N25O28S8

Molecular Weight

2346.04

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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