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SIAIS100

Product Specifications

Target

PROTACs, Others, Bcr-Abl

Related Pathways

Tyrosine Kinase/Adaptors, Others, Angiogenesis, PROTAC, Cytoskeletal Signaling

Bioactivity

SIAIS100, a potent BCR-ABL PROTAC degrader, demonstrates a DC50 value of 2.7 nM, highlighting its efficacy. It is primarily utilized in the investigation of chronic myeloid leukemia (CML) [1].

Molecular Formula

C44H50ClF2N9O5S

Molecular Weight

890.44

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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