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KRas G12R inhibitor 1

Product Specifications

Target

Others|||Kras|||Ras

Related Pathways

MAPK|||GPCR/G Protein|||Others

Bioactivity

KRas G12R Inhibitor 1 (compound 3) is a selective covalent inhibitor targeting the KRas G12R mutation, leveraging the high nucleophilicity of mutant cysteines to bind irreversibly within the K-Ras Switch II region. This compound is utilized in cancer research [1].

Molecular Formula

C39H38ClF7N6O9

Molecular Weight

903.2

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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