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LSD1-IN-26

Product Specifications

Target

Others, Monoamine Oxidase, Bcl-2 Family, Apoptosis, Caspase, Histone Demethylase, IAP

Related Pathways

Apoptosis, Chromatin/Epigenetic, Proteases/Proteasome, Neuroscience, Others

Bioactivity

LSD1-IN-26 (compound 12u), a potent LSD1 inhibitor, exhibits an IC50 of 25.3 nM. It also demonstrates inhibition of MAO-A (IC50 = 1234.57 nM) and MAO-B (IC50 = 3819.27 nM), significantly inducing apoptosis in MGC-803 cells. This compound is applicable in gastric cancer research [1].

Molecular Formula

C27H25Cl2F2N3O

Molecular Weight

516.41

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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