PROTAC CDK9 degrader-5
Product Specifications
CAS Number
2935587-89-4
Target
CDK, PROTACs
Related Pathways
PROTAC, Cell Cycle/Checkpoint
Bioactivity
PROTAC CDK9 degrader-5 is a selective PROTAC that mediates degradation of CDK9 via the proteasome pathway, efficiently degrading CDK9 42 and CDK9 55 isoforms with DC50 values of 0.10 μM and 0.14 μM, respectively [1].
Smiles
O=C1C=2C(C(=O)N1C3C(=O)NC(=O)CC3)=CC=CC2OCC(NCCCCCCCCCCC(=O)N4CCC(NC(=O)C=5C(NC(=O)C6=C(Cl)C=CC=C6Cl)=CNN5)CC4)=O
Molecular Formula
C42H48Cl2N8O9
Molecular Weight
879.78
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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