MS8815
Product Specifications
CAS Number
2855085-25-3
Target
PROTACs, Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic, PROTAC
Bioactivity
MS8815, a selective proteolysis targeting chimera (PROTAC) degrader of enhancer of zeste homolog 2 (EZH2), exhibits inhibitory activity with an IC50 value of 8.6 nM. It is utilized in the research of triple-negative breast cancer (TNBC) [1].
Smiles
CCN(C1CCOCC1)c1cc(cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)-c1ccc(CN2CCN(CC2)C(=O)CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(cc2)-c2scnc2C)C(C)(C)C)cc1
Molecular Formula
C65H87N9O8S
Molecular Weight
1154.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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