SW2_152F
Product Specifications
Target
Histone Methyltransferase, Others
Related Pathways
Chromatin/Epigenetic, Others
Bioactivity
SW2_152F is a potent and selective inhibitor of the chromobox 2 chromodomain (CBX2 ChD), exhibiting a dissociation constant (K d) of 80 nM. It demonstrates 24-1000-fold greater selectivity for CBX2 ChD over other CBX paralogs in vitro [1].
Smiles
ClC1=CC(Cl)=CC(C(N[C@@H](CC2=CC=C(O)C(Cl)=C2)C(N[C@@H](C3CCCC3)C(N[C@H]([C@@H](C)CC)C(N[C@@H](CCCCN(CC)CC)C(N[C@@H](CO)C(NCC#C)=O)=O)=O)=O)=O)=O)=C1
Molecular Formula
C45H62Cl3N7O8
Molecular Weight
935.37
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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