What is the catalog number for PROTAC BRD4 Degrader-12?

The catalog number for PROTAC BRD4 Degrader-12 is T74125.

What sizes are available for PROTAC BRD4 Degrader-12?

PROTAC BRD4 Degrader-12 is available in the following size(s): 5 mg, 50 mg.

How many pack sizes does PROTAC BRD4 Degrader-12 come in?

PROTAC BRD4 Degrader-12 is available in 2 different pack sizes.

Is PROTAC BRD4 Degrader-12 in stock?

PROTAC BRD4 Degrader-12 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures PROTAC BRD4 Degrader-12?

PROTAC BRD4 Degrader-12 is manufactured by Molfinity.

What is the estimated delivery time for PROTAC BRD4 Degrader-12?

Estimated delivery time for PROTAC BRD4 Degrader-12 is approximately 10 business day(s), depending on your location.

PROTAC BRD4 Degrader-12

Product Specifications

CAS Number

2417370-90-0

Target

Epigenetic Reader Domain, PROTAC-Linker Conjugates for PAC, PROTACs, Others

Related Pathways

PROTAC, Chromatin/Epigenetic, Antibody-drug Conjugate/ADC Related, Others

Bioactivity

PROTAC BRD4 Degrader-12 (compound 9c) is a PROTAC that links von Hippel-Lindau and BRD4 ligands. When conjugated with STEAP1 and CLL1 antibodies, this compound effectively degrades BRD4 protein in PC3 prostate cancer cells, demonstrating potent activity with DC50 values of 0.39 nM and 0.24 nM, respectively [1].

Smiles

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