Ep300/CREBBP-IN-2
Product Specifications
CAS Number
2259641-59-1
Target
Others|||Histone Acetyltransferase
Related Pathways
Chromatin/Epigenetic|||Others
Bioactivity
Ep300/CREBBP-IN-2 (Example 73) is a potent, orally bioavailable inhibitor of Ep300 and CREBBP, with IC50 values of 0.052 ?M and 0.148 ?M, respectively, and is used in cancer research [1].
Smiles
COc1ccc(cc1)C1(CCC(F)(F)CC1)C(=O)N1C[C@H](F)C[C@@H]1C(=O)Nc1ccc2NC(=O)Cc2n1
Molecular Formula
C26H27F3N4O4
Molecular Weight
516.51
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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