ARL67156 triethylamine
Product Specifications
Target
Others, Phosphatase
Related Pathways
Metabolism, Others
Bioactivity
ARL67156 (FPL 67156) triethylamine, a selective ecto-ATPase inhibitor, functions as a competitive inhibitor for NTPDase1 (CD39), NTPDase3, and NPP1, exhibiting inhibition constants (Kis) of 11, 18, and 12 μM, respectively. This compound is applicable in researching diseases such as calcific aortic valve disease and asthma [1] [2].
Molecular Formula
C15H24Br2N5O12P3. (4.3C6H15N)
Molecular Weight
1154.23
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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