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RX 801077

Product Specifications

CAS Number

72583-92-7

Target

Others|||Imidazoline Receptor

Related Pathways

Others|||Neuroscience

Bioactivity

RX 801077 (2 BFI free base), a selective imidazoline I2 receptor (I2R) agonist with a K_i value of 70.1 nM, demonstrates anti-inflammatory and neuroprotective properties, making it a potential research candidate for traumatic brain injury (TBI) .

Smiles

C1(=CC=2C(O1)=CC=CC2)C=3NCCN3

Molecular Formula

C11H10N2O

Molecular Weight

186.21

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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