(S) -HH2853
Product Specifications
CAS Number
2202678-05-3
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9974
Bioactivity
(S) -HH2853 is a potent dual inhibitor of EZH1 and EZH2, inhibiting EZH2_Y641F with an IC50 of <100 nM. (S) -HH2853 has potential antitumor activity and can be used in the study of autoimmune diseases.
Smiles
[C@H](C)(C=1N2C(=C(C=C2)C3=CC=C(C)N=N3)C=C(C(NCC4=C(OC)C=C(C)NC4=O)=O)C1C)N5CCN(CC(F)(F)F)CC5
Molecular Formula
C31H36F3N7O3
Molecular Weight
611.66
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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