BAY 1214784
Product Specifications
CAS Number
1631164-25-4
Target
Others, GNRH Receptor
Related Pathways
GPCR/G Protein, Others
Purity
1
Bioactivity
BAY 1214784, a potent, selective, and orally active spiroindoline derivative compound, serves as an antagonist of the human gonadotropin-releasing hormone receptor (hGnRH-R) . It notably reduces plasma luteinizing hormone levels by up to 49%, demonstrating low pharmacokinetic variability and good tolerability. This compound shows promise for research into uterine fibroids.
Smiles
S(=O)(=O)(N1[C@@H](C2(C=3C1=CC=C(C(NCC4=C(Cl)C=C(C(F)(F)F)C=N4)=O)C3)CCS(=O)(=O)CC2)[C@@H]5CC5)C6=CC=C(F)C=C6
Molecular Formula
C29H26ClF4N3O5S2
Molecular Weight
672.11
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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