Palazestrant
Product Specifications
CAS Number
2092925-89-6
Target
Estrogen/progestogen Receptor, Estrogen Receptor/ERR
Related Pathways
Endocrinology/Hormones
Purity
0.9755
Bioactivity
Palazestrant (OP-1250) is an orally available and highly potent estrogen receptor antagonist and selective ER degrader with antitumor activity.Palazestrant inhibits 17b-estradiol (E2), inhibits MCF7 and CAMA-1 cell proliferation, and can be used in breast cancer research.
Smiles
C(C(C)(C)F)N1[C@@H](C2=C(C=3C(N2)=CC=CC3)C[C@H]1C)C4=CC=C(OC5CN(CCC)C5)C=C4
Molecular Formula
C28H36FN3O
Molecular Weight
449.6
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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