PKCiota-IN-1
Product Specifications
CAS Number
2230052-97-6
Target
Others, PKC
Related Pathways
Others, Cytoskeletal Signaling, Chromatin/Epigenetic
Bioactivity
PKCiota-IN-1 is a potent inhibitor of PKCiota (PKC-ι), exhibiting an IC50 of 2.7 nM. Additionally, it displays inhibitory activity against PKC-α and PKC-ε, with IC50 values of 45 nM and 450 nM, respectively.
Smiles
O(C)C1=C(C2=C3N(N=C2)C=CC(=C3)C4=C5C(=NC=C4)NC=C5)C=C6C(=C1)CC(CF)NC6
Molecular Formula
C25H22FN5O
Molecular Weight
427.47
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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