Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

PARP-2/1-IN-2

Product Specifications

CAS Number

912444-01-0

Target

Others|||PARP

Related Pathways

DNA Damage/DNA Repair|||Chromatin/Epigenetic|||Others

Bioactivity

PARP-2/1-IN-2, an enantiomer of Veliparib, serves as a potent inhibitor of PARP, demonstrating inhibition constants (Kis) of 2 nM for PARP-2 and 5 nM for PARP-1. This compound exhibits a half-maximal effective concentration (EC50) of 3 nM in cell-based assays evaluating PARP activity [1].

Smiles

C(N)(=O)C1=C2C(N=C(N2)[C@]3(C)CCCN3)=CC=C1

Molecular Formula

C13H16N4O

Molecular Weight

244.29

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

Lentiviral human CACNA2D2 shRNA (UAS) - Lentiviral human CACNA2D2 shRNA (UAS, iRFP) (100)
GTR15148935 1 Vial

Lentiviral human CACNA2D2 shRNA (UAS) - Lentiviral human CACNA2D2 shRNA (UAS, iRFP) (100)

Ask
View Details
S100A9 (Biotin)
575504-01 50 µg

S100A9 (Biotin)

Ask
View Details
S100A9 (Biotin)
575504-02 100 µg

S100A9 (Biotin)

Ask
View Details
Mmu-miR-7022-5p mimic
HY-R03781-01 5 nmol

Mmu-miR-7022-5p mimic

Ask
View Details
Mmu-miR-7022-5p mimic
HY-R03781-02 20 nmol

Mmu-miR-7022-5p mimic

Ask
View Details
DYRK3 Polyclonal Antibody, FITC Conjugated
bs-9520R-FITC 100 µL

DYRK3 Polyclonal Antibody, FITC Conjugated

Ask
View Details