PBRM1-BD2-IN-1
Product Specifications
CAS Number
1915012-21-3
Target
Others|||Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic|||Others
Bioactivity
PBRM1-BD2-IN-1 is a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, exhibiting a binding affinity (Kd) of 0.7 ?M and an inhibitory efficacy (IC50) of 0.2 ?M, and is used in cancer research.
Smiles
C(\C(CC)CC)=C\1/C=2N(C=3C(C(=O)N2)=C(Cl)C=CC3)CC1
Molecular Formula
C17H19ClN2O
Molecular Weight
302.8
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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