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BRD4 Inhibitor-25

Product Specifications

Target

Others, Epigenetic Reader Domain

Related Pathways

Others, Chromatin/Epigenetic

Bioactivity

BRD4 Inhibitor-25, a chemical compound targeting the BD1 and BD2 domains of BRD4 with half-maximal inhibitory concentrations (IC50s) of 0.82 μM and 1.94 μM respectively, demonstrates efficacy in inducing apoptotic and autophagic cell death in ovarian cancer cells. This compound is utilized in researching cancers, cardiovascular, neuromuscular, and inflammatory disorders.

Molecular Formula

C29H27N5O6S

Molecular Weight

573.62

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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