GnRH-R antagonist 1
Product Specifications
CAS Number
2826273-90-7
Target
GNRH Receptor
Related Pathways
GPCR/G Protein
Bioactivity
GnRH-R antagonist 1 (Compound 21a), is an orally active, membrane-permeable agent with a high binding affinity (IC50=0.57 nM) and potent in vitro antagonistic efficacy (IC50=2.18 nM) . It is utilized in research focused on advanced prostate cancer and the prevention of premature LH surges [1].
Smiles
CN(CCOC(F)(F)F)CC1=C(SC2=C1C(=O)N(C(=O)N2CC3=C(C=CC=C3F)F)C4=NN=C(C=C4)OC)C5=CC=C(C=C5)NC(=O)NOC
Molecular Formula
C31H28F5N7O6S
Molecular Weight
721.65
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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