PF-4348235 HCl
Product Specifications
Target
AChR|||Adrenergic Receptor
Related Pathways
GPCR/G Protein|||Neuroscience
Purity
0.9966
Bioactivity
PF-4348235 HCl (?2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and ?2 adrenergic receptor agonist (MABA, EC50: 3.7 nM) . PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD) .
Smiles
O[C@H](C1=CC(NS(C)(=O)=O)=C(C=C1)O)CNCCCCCCCCCN(CC2)CCC2OC(NC3=C(C4=CC(Cl)=C(C=C4)O)C=CC=C3)=O.Cl
Molecular Formula
C36H50Cl2N4O7S
Molecular Weight
753.78
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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