DSP-1053 benzenesulfonate
Product Specifications
CAS Number
1176326-78-5
Target
5-HT Receptor|||Serotonin Transporter|||Others
Related Pathways
GPCR/G Protein|||Neuroscience|||Others
Bioactivity
DSP-1053, a benzylpiperidine derivative, is a potent serotonin transporter (SERT) inhibitor with a dissociation constant (K_i) of 1.02 nM and exhibits partial agonistic activity at the 5-HT_1A receptor with a K_i of 5.05 nM, indicating its potential as an antidepressant.
Smiles
O=C1C2=CC(=CC=C2OCC1)CCN3CCC(CC4=CC=C(Br)C(OCCOC)=C4)CC3.O=S(=O)(O)C=1C=CC=CC1
Molecular Formula
C32H38BrNO7S
Molecular Weight
660.62
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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