Lesogaberan hydrochloride
Product Specifications
Target
Others
Related Pathways
Others
Bioactivity
Lesogaberan (AZD-3355) hydrochloride is a potent and selective GABA B receptor agonist with an EC 50 of 8.6 nM for human recombinant GABA B receptor. The affinity (K i s) of Lesogaberan hydrochloride for rat GABA B and GABA A receptors, as measured by displacement of GABA binding in brain membranes: 5.1 nM and 1.4 ?M, respectively. Lesogaberan hydrochloride inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action .
Smiles
F[C@@H](CP(O)([H])=O)CN.Cl
Molecular Formula
C3H10ClFNO2P
Molecular Weight
177.54
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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