YM-58790
Product Specifications
CAS Number
168830-70-4
Target
AChR
Related Pathways
Neuroscience
Purity
0.9987
Bioactivity
YM-58790 free base is a potent mAChR antagonist that inhibits M1 mAChR, M2 mAChR, and M3 mAChR with Ki values of 28 nM, 260 nM, and 15 nM, respectively. It inhibits reflex rhythmic bladder contractions in rats by inhibiting bladder pressurization.
Smiles
C(NC(OC1CCN(CC2=CC=C(NC)C=C2)CC1)=O)(C3=CC=CC=C3)C4=CC=CC=C4
Molecular Formula
C27H31N3O2
Molecular Weight
429.55
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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