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ML-077

Product Specifications

CAS Number

1135304-61-8

Target

Others

Related Pathways

Others

Bioactivity

ML-077, also known as VU0255011, is a highly selective, potent, saline soluble, best in class" KCC2 antagonist for high fidelity in vitro studies on KCC2 function with IC (50) =537 nM. ML-077 is cell permeable and exhibits submicromolar potency

Smiles

CN(C(=O)CSc1ccc(nn1)-c1ccccc1)c1nc(C)cs1

Molecular Formula

C17H16N4OS2

Molecular Weight

356.47

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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