(±) -C3001a
Product Specifications
CAS Number
1374325-56-0
Target
Others, Potassium Channel
Related Pathways
Membrane transporter/Ion channel, Others
Purity
0.9913
Bioactivity
(±) -C3001a is the racemic mixture of C3001a (CAS: 2415154-29-7) . C3001a is a selective activator of the TREK channel within the two-pore-domain potassium channel (K2P) family. C3001a specifically binds to a cryptic site formed by P1 and TM4 in TREK-1, thereby promoting the selective regulation of TREK-1 activity. C3001a targets TREK channels in the peripheral nervous system, reducing the excitability of pain-sensing neurons.
Smiles
O=C(O)C1CCC(C(=O)NC2=CC=C(C=C2)C3=NC=4C=CC(=CC4S3)C)C1
Molecular Formula
C21H20N2O3S
Molecular Weight
380.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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