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PF-04671536

Product Specifications

CAS Number

1305116-69-1

Target

PDE|||Others

Related Pathways

Metabolism|||Others

Bioactivity

PF-04671536 is a highly potent and selective inhibitor of phosphodiesterase 8B (PDE8B) phosphodiesterase 8A (PDE8A) . In primary human pancreatic islets, PF-04671536 increases insulin secretion in a glucose-dependent manner.

Smiles

C(N1C=2C(N=N1)=C(N)N=C(C)N2)[C@H]3CN(CC4=NC=CS4)CCO3

Molecular Formula

C14H18N8OS

Molecular Weight

346.41

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/D16B3B30-5390-41B8-BE23-4000D54FF160/T71020

Available Sizes

Curated Selection

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