PF-04671536
Product Specifications
CAS Number
1305116-69-1
Target
PDE, Others
Related Pathways
Metabolism, Others
Bioactivity
PF-04671536 is a highly potent and selective inhibitor of phosphodiesterase 8B (PDE8B) phosphodiesterase 8A (PDE8A) . In primary human pancreatic islets, PF-04671536 increases insulin secretion in a glucose-dependent manner.
Smiles
C(N1C=2C(N=N1)=C(N)N=C(C)N2)[C@H]3CN(CC4=NC=CS4)CCO3
Molecular Formula
C14H18N8OS
Molecular Weight
346.41
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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