PT-S58
Product Specifications
CAS Number
1356497-92-1
Target
Others, PPAR
Related Pathways
Metabolism, Others, DNA Damage/DNA Repair
Bioactivity
PT-S58 is a PPAR β/δ full antagonist, and a derivative of GSK0660. PT-S58 has a three-fold higher affinity for the receptor than GSK0660 and is a potent inhibitor of agonist-induced target gene expression. PT-S58 are effective on PPRE-independent functions of PPARβ/δ. Unlike GSK0660, PT-S58 blocks the recruitment co-repressor molecules such as SMRT.
Smiles
S(NC1=C(OC)C=C(NC(C)(C)C)C=C1)(=O)(=O)C2=C(C(OC)=O)SC=C2
Molecular Formula
C17H22N2O5S2
Molecular Weight
398.5
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
TRV-0020031-01 50 Tests
Anti-Sex Hormone Binding Globulin (SHBG) Monoclonal Antibody
Sign In for Pricing
View Details TRV-0020031-02 100 Tests
Anti-Sex Hormone Binding Globulin (SHBG) Monoclonal Antibody
Sign In for Pricing
View Details TRV-0020031-03 200 Tests
Anti-Sex Hormone Binding Globulin (SHBG) Monoclonal Antibody
Sign In for Pricing
View Details VAng-Lsx9998-500gEcoli 500 µg (E. coli)
Recombinant Clostridium Novyi ispE Protein (aa 1-280)
Sign In for Pricing
View Details 