Rimegepant sulfate hydrate
Product Specifications
CAS Number
1374024-48-2
Target
CGRP Receptor, Others
Related Pathways
Others, Neuroscience, GPCR/G Protein
Bioactivity
Rimegepant, also known as BMS-927711 and BHV-3000, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines. Rimegepant has shown in vivo efficacy without vasoconstriction effect. BMS-927711 is superior to placebo at several different doses (75 mg, 150 mg, and 300 mg) and has an excellent tolerability profile.
Smiles
O.OS(O)(=O)=O.N[C@H]1[C@@H](CC[C@@H](OC(=O)N2CCC(CC2)n2c3cccnc3[nH]c2=O)c2ncccc12)c1cccc(F)c1F
Molecular Formula
C56H64F4N12O13S
Molecular Weight
1221.2526
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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