Rimegepant sulfate hydrate
Product Specifications
CAS Number
1374024-48-2
Target
CGRP Receptor, Others
Related Pathways
Others, Neuroscience, GPCR/G Protein
Bioactivity
Rimegepant, also known as BMS-927711 and BHV-3000, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines. Rimegepant has shown in vivo efficacy without vasoconstriction effect. BMS-927711 is superior to placebo at several different doses (75 mg, 150 mg, and 300 mg) and has an excellent tolerability profile.
Smiles
O.OS(O)(=O)=O.N[C@H]1[C@@H](CC[C@@H](OC(=O)N2CCC(CC2)n2c3cccnc3[nH]c2=O)c2ncccc12)c1cccc(F)c1F
Molecular Formula
C56H64F4N12O13S
Molecular Weight
1221.2526
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
BNC403291-100 1x 100 µL
Sarcomeric Actinin Alpha 2 / ACTN2 (ACTN2/3291), CF640R conjugate, 0.1mg/mL
Sign In for Pricing
View Details ![RHOJ Mouse Monoclonal Antibody (HRP conjugated) [Clone ID: OTI5E5]](https://cdn.genprice.uk/products/937/68dd1b70061270361ea18230/imageurl/ta505595bm.webp)
TA505595BM 100 µL
RHOJ Mouse Monoclonal Antibody (HRP conjugated) [Clone ID: OTI5E5]
Sign In for Pricing
View Details 
RDR-TMEM27-Hu-01 96 Tests
Human Transmembrane Protein 27 (TMEM27) ELISA Kit
Sign In for Pricing
View Details RDR-TMEM27-Hu-02 48 Tests
Human Transmembrane Protein 27 (TMEM27) ELISA Kit
Sign In for Pricing
View Details 