GAT100
Product Specifications
CAS Number
1663564-42-8
Target
Others
Related Pathways
Others
Bioactivity
GAT100 is a potent and covalent negative allosteric modulator (NAM) . GAT-100 behaved as a robust positive allosteric modulator of binding of orthosteric agonist CP55,940. This novel covalent probe can serve as a useful tool for characterizing CB1R allosteric ligand-binding motifs.
Smiles
C(C)C=1C=2C(NC1C(NCCC3=CC=C(C=C3)N4CCCCC4)=O)=CC=C(N=C=S)C2
Molecular Formula
C25H28N4OS
Molecular Weight
432.58
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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