Tasimelteon-d5
Product Specifications
CAS Number
1962124-51-1
Target
Melatonin Receptor
Related Pathways
GPCR/G Protein
Bioactivity
Tasimelteon-d5 is intended for use as an internal standard for the quantification of tasimelteon by GC- or LC-MS. Tasimelteon is a melatonin (MT) receptor agonist. It selectively binds MT1 and MT2 receptors over a panel of 160 additional receptors and enzymes at 10 μM. Tasimelteon inhibits forskolin-induced cAMP accumulation with EC50 values of 0.79 and 1 nM in NIH3T3 cells expressing the MT1 or MT2 receptor, respectively. Formulations containing tasimelteon have been used in the treatment of non-24-hour sleep-wake disorder.
Smiles
C(NC(C(C([2H])([2H])[2H])([2H])[2H])=O)[C@H]1[C@@H](C1)C2=C3C(=CC=C2)OCC3
Molecular Formula
C15H14D5NO2
Molecular Weight
250.35
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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