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EPZ020411 HCl

Product Specifications

CAS Number

2095432-47-4

Target

Others

Related Pathways

Others

Bioactivity

EPZ020411 is a potent and selective PRMT6 inhibitor tool compound. EPZ020411 shows good bioavailability following subcutaneous dosing in rats making it a suitable tool for in vivo studies. EPZ020411 suppresses RCC1 arginine methylation and improves the cytotoxic activity of radiotherapy against GSC brain tumor xenografts.

Smiles

C(N(CCNC)C)C=1C(=NNC1)C2=CC=C(O[C@H]3C[C@H](OCCC4CCOCC4)C3)C=C2.Cl.Cl

Molecular Formula

C25H40Cl2N4O3

Molecular Weight

515.52

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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